Skip to main content
Go to the home page of the European Commission (opens in new window)
English en
CORDIS - EU research results
CORDIS
Content archived on 2024-05-29

The development of a modular approach to stereocontrolled oligosaccharide synthesis by intramolecular glycosylation

Objective

It is now well established that oligosaccharides play fundamental roles in an enormously wide range of important biological processes, including viral and bacterial infectivity, antigenicity and cancer metastasis. In addition it also now recognized that th e post-translational modification of proteins by glycosylation plays a crucial role in successful protein folding, and on the conformation, metabolic stability and catalytic activity of folded glycoproteins. However in the vast majority of cases the functi on of the oligosaccharide is not yet precisely understood, and there is a need for synthetic oligosaccharides in order to elucidate the roles that these oligomers play in their varied environments. Despite impressive recent developments, no synthetic metho dology currently exists that allows the synthesis of oligosaccharides in a reliable and generally applicable manner. The research program we propose will centre on the further development of novel synthetic methodology for construction of synthetic oligosa ccharides, crucially in a totally stereoselective and potentially automatable fashion. The proposal centres on the development of a modular approach to sterecontrolled oligosaccharide synthesis. The crucial point is that whilst neighbouring group participa tion will be employed to give 1,2-trans glycosidic linkages using standard intermolecular glycosylation reactions, that by actually using the same building blocks we shall be able to achieve the stereoselective synthesis of 1,2-cis glycosidic linkages simp ly by performing intramolecular glycosylation reactions. Importantly both sets of reaction conditions will involve the same component steps, but by performing each of these individual steps in a different order we will be able to totally control the stereo chemical outcome of the glycosylation reaction. Such an approach would allow the development of the first oligosaccharide synthesiser wherein the problem of anomeric stereocontrol had been truly addressed.

Fields of science (EuroSciVoc)

CORDIS classifies projects with EuroSciVoc, a multilingual taxonomy of fields of science, through a semi-automatic process based on NLP techniques. See: The European Science Vocabulary.

You need to log in or register to use this function

Topic(s)

Calls for proposals are divided into topics. A topic defines a specific subject or area for which applicants can submit proposals. The description of a topic comprises its specific scope and the expected impact of the funded project.

Call for proposal

Procedure for inviting applicants to submit project proposals, with the aim of receiving EU funding.

FP6-2002-MOBILITY-5
See other projects for this call

Funding Scheme

Funding scheme (or “Type of Action”) inside a programme with common features. It specifies: the scope of what is funded; the reimbursement rate; specific evaluation criteria to qualify for funding; and the use of simplified forms of costs like lump sums.

EIF - Marie Curie actions-Intra-European Fellowships

Coordinator

CHANCELLOR, MASTERS AND SCHOLARS OF THE UNIVERSITY OF OXFORD
EU contribution
No data
Address
University Offices, Wellington Square
OXFORD
United Kingdom

See on map

Links
Total cost

The total costs incurred by this organisation to participate in the project, including direct and indirect costs. This amount is a subset of the overall project budget.

No data
My booklet 0 0