PROTAC Linker Design: towards Functionality

Project Information

PREDICT

Grant agreement ID: 101026833

DOI

10.3030/101026833

Project closed

EC signature date 23 March 2021

Start date 1 July 2021

End date 30 June 2023

Funded under

• EXCELLENT SCIENCE - Marie Skłodowska-Curie Actions

Total cost

€ 212 933,76

EU contribution

€ 212 933,76

Coordinated by

UNIVERSITY OF DUNDEE
United Kingdom

CORDIS provides links to public deliverables and publications of HORIZON projects.

Links to deliverables and publications from FP7 projects, as well as links to some specific result types such as dataset and software, are dynamically retrieved from OpenAIRE .

Publications

Peer reviewed articles (1)

Discovery of small molecule ligands for the von Hippel-Lindau (VHL) E3 ligase and their use as inhibitors and PROTAC degraders

Author(s): Claudia J. Diehl, Alessio Ciulli
Published in: Chemical Society Reviews, Issue 51, 2022, Page(s) 8216-8257, ISSN 0306-0012
Publisher: Royal Society of Chemistry
DOI: 10.1039/d2cs00387b

Non-peer reviewed articles (1)

Expanding the Structural Diversity at the Phenylene Core of Ligands for the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase: Development of Highly Potent Hypoxia-Inducible Factor-1alpha (HIF-1alpha) Stabilizers

Author(s): Lan Phuong Vu, Claudia J. Diehl, Ryan Casement, Adam Bond, Christian Steinebach, Nika Strasek, Alesa Bricelj, Andrej Perdih, Gregor Schnakenburg, Izidor Sosic, Alessio Ciulli Author, Michael Gutschow
Published in: ChemRxiv, 2023, ISSN 2573-2293
Publisher: Cambridge Open Engage
DOI: 10.26434/chemrxiv-2023-5gbb6-v2