Fast Quantitative Validation of 3D Models of Low-Affinity Protein–Ligand Complexes by STD NMR Spectroscopy
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Author(s):
Ridvan Nepravishta, Jonathan Ramírez-Cárdenas, Gabriel Rocha, Samuel Walpole, Thomas Hicks, Serena Monaco, Juan C. Muñoz-García, Jesús Angulo
Published in:
Journal of Medicinal Chemistry, 2024, ISSN 1520-4804
Publisher:
American Chemical Society
DOI:
10.1021/acs.jmedchem.4c00204
Speeding-up the Determination of Protein–Ligand Affinities by STD NMR: The Reduced Data Set STD NMR Approach (rd-STD NMR)
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Author(s):
Gabriel Rocha, Jonathan Ramírez-Cárdenas, M. Carmen Padilla-Pérez, Samuel Walpole, Ridvan Nepravishta, M. Isabel García-Moreno, Elena M. Sánchez-Fernández, Carmen Ortiz Mellet, Jesús Angulo*, and Juan C. Muñoz-García*
Published in:
Analytical Chemistry, ISSN 1520-6882
Publisher:
American Chemical Society
DOI:
10.1021/ACS.ANALCHEM.3C03980