The CDK inhibitor CR8 acts as a molecular glue degrader that depletes cyclin K
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Author(s):
Mikołaj Słabicki, Zuzanna Kozicka, Georg Petzold, Yen-Der Li, Manisha Manojkumar, Richard D. Bunker, Katherine A. Donovan, Quinlan L. Sievers, Jonas Koeppel, Dakota Suchyta, Adam S. Sperling, Emma C. Fink, Jessica A. Gasser, Li R. Wang, Steven M. Corsello, Rob S. Sellar, Max Jan, Dennis Gillingham, Claudia Scholl, Stefan Fröhling, Todd R. Golub, Eric S. Fischer, Nicolas H. Thomä, Benjamin L. E
Published in:
Nature, Issue 585/7824, 2020, Page(s) 293-297, ISSN 0028-0836
Publisher:
Nature Publishing Group
DOI:
10.1038/s41586-020-2374-x
Defining the human C2H2 zinc finger degrome targeted by thalidomide analogs through CRBN
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Author(s):
Quinlan L. Sievers, Georg Petzold, Richard D. Bunker, Aline Renneville, Mikołaj Słabicki, Brian J. Liddicoat, Wassim Abdulrahman, Tarjei Mikkelsen, Benjamin L. Ebert, Nicolas H. Thomä
Published in:
Science, Issue 362/6414, 2018, Page(s) eaat0572, ISSN 0036-8075
Publisher:
American Association for the Advancement of Science
DOI:
10.1126/science.aat0572
Small-molecule-induced polymerization triggers degradation of BCL6
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Author(s):
Mikołaj Słabicki, Hojong Yoon, Jonas Koeppel, Lena Nitsch, Shourya S. Roy Burman, Cristina Di Genua, Katherine A. Donovan, Adam S. Sperling, Moritz Hunkeler, Jonathan M. Tsai, Rohan Sharma, Andrew Guirguis, Charles Zou, Priya Chudasama, Jessica A. Gasser, Peter G. Miller, Claudia Scholl, Stefan Fröhling, Radosław P. Nowak, Eric S. Fischer, Benjamin L. Ebert
Published in:
Nature, Issue 588/7836, 2020, Page(s) 164-168, ISSN 0028-0836
Publisher:
Nature Publishing Group
DOI:
10.1038/s41586-020-2925-1