Non-Natural Linker Configuration in 2,6-Dipeptidyl-Anthraquinones Enhances the Inhibition of TAR RNA Binding/Annealing Activities by HIV-1 NC and Tat Proteins
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Author(s):
Alice Sosic, Irene Saccone, Caterina Carraro, Thomas Kenderdine, Elia Gamba, Giuseppe Caliendo, Angela Corvino, Paola Di Vaio, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Beatrice Severino, Valentina Spada, Dan Fabris, Francesco Frecentese, Barbara Gatto
Published in:
Bioconjugate Chemistry, Issue 29/7, 2018, Page(s) 2195-2207, ISSN 1043-1802
Publisher:
American Chemical Society
DOI:
10.1021/acs.bioconjchem.8b00104
Behind the Mirror: Chirality Tunes the Reactivity and Cytotoxicity of Chloropiperidines as Potential Anticancer Agents
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Author(s):
Caterina Carraro, Alexander Francke, Alice Sosic, Franziska Kohl, Tim Helbing, Michele De Franco, Daniele Fabris, Richard Göttlich, Barbara Gatto
Published in:
ACS Medicinal Chemistry Letters, Issue 10/4, 2019, Page(s) 552-557, ISSN 1948-5875
Publisher:
American Chemical Society
DOI:
10.1021/acsmedchemlett.8b00580