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Overcoming the Selectivity Challenge in Chemistry and Chemical Biology via Innovative Tethering Strategies

Deliverables

Data Management Plan

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Publications

Palladium-Catalyzed Functionalization of Olefins and Alkynes: From Oxyalkynylation to Tethered Dynamic Kinetic Asymmetric Transformations (DYKAT)

Author(s): Stefano Nicolai, Ugo Orcel, Bastian Muriel, Phillip D. G. Greenwood, Luca Buzzetti, Mikus Puriņš, Jerome Waser
Published in: Synlett, 2021, Page(s) 472-487, ISSN 0936-5214
DOI: 10.1055/a-1308-0021

Cys–Cys and Cys–Lys Stapling of Unprotected Peptides Enabled by Hypervalent Iodine Reagents

Author(s): Javier Ceballos, Elija Grinhagena, Gontran Sangouard, Christian Heinis, Jerome Waser
Published in: Angewandte Chemie International Edition, Issue 60/16, 2021, Page(s) 9022-9031, ISSN 1433-7851
DOI: 10.1002/anie.202014511

Enantioselective Carboetherification/Hydrogenation for the Synthesis of Amino Alcohols via a Catalytically Formed Chiral Auxiliary

Author(s): Luca Buzzetti, Mikus Puriņš, Phillip D. G. Greenwood, Jerome Waser
Published in: Journal of the American Chemical Society, Issue 142/41, 2020, Page(s) 17334-17339, ISSN 0002-7863
DOI: 10.1021/jacs.0c09177

Palladium-Catalyzed Carboxy-Alkynylation of Propargylic Amines Using Carbonate Salts as Carbon Dioxide Source

Author(s): Phillip D. G. Greenwood, Jerome Waser
Published in: European Journal of Organic Chemistry, Issue 2019/31-32, 2019, Page(s) 5183-5186, ISSN 1434-193X
DOI: 10.1002/ejoc.201900500

“Doubly Orthogonal” Labeling of Peptides and Proteins

Author(s): Romain Tessier, Javier Ceballos, Nora Guidotti, Raphael Simonet-Davin, Beat Fierz, Jerome Waser
Published in: Chem, Issue 5/8, 2019, Page(s) 2243-2263, ISSN 2451-9294
DOI: 10.1016/j.chempr.2019.06.022

Ethynylation of Cysteine Residues: From Peptides to Proteins in Vitro and in Living Cells

Author(s): Romain Tessier, Raj Kumar Nandi, Brendan G. Dwyer, Daniel Abegg, Charlotte Sornay, Javier Ceballos, Stéphane Erb, Sarah Cianférani, Alain Wagner, Guilhem Chaubet, Alexander Adibekian, Jerome Waser
Published in: Angewandte Chemie International Edition, Issue 59/27, 2020, Page(s) 10961-10970, ISSN 1433-7851
DOI: 10.1002/anie.202002626

Amphiphilic Iodine(III) Reagents for the Lipophilization of Peptides in Water

Author(s): Abhaya Kumar Mishra, Romain Tessier, Durga Prasad Hari, Jerome Waser
Published in: Angewandte Chemie International Edition, Issue 60/33, 2021, Page(s) 17963-17968, ISSN 1433-7851
DOI: 10.1002/anie.202106458

Inhibition of Thiol‐Mediated Uptake with Irreversible Covalent Inhibitors

Author(s): Bumhee Lim, Yangyang Cheng, Takehiro Kato, Anh‐Tuan Pham, Eliott Le Du, Abhaya Kumar Mishra, Elija Grinhagena, Dimitri Moreau, Naomi Sakai, Jerome Waser, Stefan Matile
Published in: Helvetica Chimica Acta, 2021, ISSN 0018-019X
DOI: 10.1002/hlca.202100085