Albumin-Mediated Drug Uptake by Organic Anion Transporter 1/3 Is Real: Implications for the Prediction of Active Renal Secretion Clearance
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Author(s):
Shawn Pei Feng Tan, Annika Tillmann, Susan J. Murby, Amin Rostami-Hodjegan, Daniel Scotcher, Aleksandra Galetin
Published in:
Molecular Pharmaceutics, Issue 21, 2024, Page(s) 4603-4617, ISSN 1543-8384
Publisher:
American Chemical Society
DOI:
10.1021/acs.molpharmaceut.4c00504
QSPRpred: a Flexible Open-Source Quantitative Structure-Property Relationship Modelling Tool
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Author(s):
Helle W. van den Maagdenberg, Martin Šícho, David Alencar Araripe, Sohvi Luukkonen, Linde Schoenmaker, Michiel Jespers, Olivier J. M. Béquignon, Marina Gorostiola González, Remco L. van den Broek, Andrius Bernatavicius, J. G. Coen van Hasselt, Piet. H. van der Graaf, Gerard J. P. van Westen
Published in:
Journal of Cheminformatics, Issue 16, 2024, ISSN 1758-2946
Publisher:
Chemistry Central
DOI:
10.1186/s13321-024-00908-y
Label-free but still constrained: Assessment of global proteomic strategies for the quantification of hepatic enzymes and transporters
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Author(s):
Barber J, Al-Majdoub ZM, Couto N, Vasilogianni AM, Tillmann A, Alrubia S, Rostami-Hodjegan A, Achour B.
Published in:
Drug metabolism and disposition, Issue 50, 2022, Page(s) 762-769, ISSN 0090-9556
Publisher:
American Society for Pharmacology and Experimental Therapeutics
DOI:
10.1124/dmd.121.000780
Targeting Kidney Fibrosis with Polymeric Nanocarriers
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Author(s):
Vedangi Kulkarni, Tim Caspers, Diana Moeckel, Susanne Koletnik, Elena Rama, Paraskevi Sotiropoulou, Daniel R. Dietrich, Robert Pola, Lenka Kotrchová, Tomáš Etrych, Yvonne H. W. Derks, Peter Boor, Fabian Kiessling, Felix M. Mottaghy, Barbara M. Klinkhammer, Twan Lammers
Published in:
Chemistry of Materials, Issue 36, 2024, Page(s) 9686-9695, ISSN 0897-4756
Publisher:
American Chemical Society
DOI:
10.1021/acs.chemmater.4c01788