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Photoswitchable amphiphilic lipids: a photopharmacology strategy to combat drug-resistant bacterial infections.

Publications

Tapping into the antitubercular potential of 2,5-dimethylpyrroles: A structure-activity relationship interrogation

Author(s): Dorothy Semenya Meir Touitou Domiziana Masci Camila Maringolo Ribeiro Fernando Rogerio Pavan Guilherme Felipe Dos Santos Fernandes Beatrice Gianibbi Fabrizio Manetti Daniele Castagnolo
Published in: European Journal of Medicinal Chemistry, Issue 1, 2022, ISSN 0223-5234
Publisher: Elsevier BV
DOI: 10.1016/j.ejmech.2022.114404

Oxazolidinones as versatile scaffolds in medicinal chemistry

Author(s): Guilherme Felipe Santos Fernandes Cauê Benito Scarim Seong-Heun Kim Jingyue Wu Daniele Castagnolo
Published in: RSC Medicinal Chemistry, Issue 14, 2023, Page(s) 823-847, ISSN 2632-8682
Publisher: Royal Society of Chemistry
DOI: 10.1039/d2md00415a

Tuberculosis Drug Discovery: Challenges and New Horizons

Author(s): Guilherme F. S. Fernandes Andrew M. Thompson Daniele Castagnolo William A. Denny Jean L. Dos Santos
Published in: Journal of Medicinal Chemistry, Issue 65, 2022, Page(s) 7489–7531, ISSN 0022-2623
Publisher: American Chemical Society
DOI: 10.1021/acs.jmedchem.2c00227

Development of Novel Membrane Disrupting Lipoguanidine Compounds Sensitizing Gram-Negative Bacteria to Antibiotics

Author(s): Seong-Heun Kim Charlotte K. Hind Guilherme F. S. Fernandes Jingyue Wu Dorothy Semenya Melanie Clifford Caleb Marsh Silvia Anselmi A. James Mason Kenneth D. Bruce J. Mark Sutton Daniele Castagnolo
Published in: ACS Medicinal Chemistry Letters, 2024, ISSN 1948-5875
Publisher: American Chemical Society
DOI: 10.1021/acsmedchemlett.3c00460

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