Tapping into the antitubercular potential of 2,5-dimethylpyrroles: A structure-activity relationship interrogation
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Author(s):
Dorothy Semenya
Meir Touitou
Domiziana Masci
Camila Maringolo Ribeiro
Fernando Rogerio Pavan
Guilherme Felipe Dos Santos Fernandes
Beatrice Gianibbi
Fabrizio Manetti
Daniele Castagnolo
Published in:
European Journal of Medicinal Chemistry, Issue 1, 2022, ISSN 0223-5234
Publisher:
Elsevier BV
DOI:
10.1016/j.ejmech.2022.114404
Oxazolidinones as versatile scaffolds in medicinal chemistry
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Author(s):
Guilherme Felipe Santos Fernandes
Cauê Benito Scarim
Seong-Heun Kim
Jingyue Wu
Daniele Castagnolo
Published in:
RSC Medicinal Chemistry, Issue 14, 2023, Page(s) 823-847, ISSN 2632-8682
Publisher:
Royal Society of Chemistry
DOI:
10.1039/d2md00415a
Tuberculosis Drug Discovery: Challenges and New Horizons
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Author(s):
Guilherme F. S. Fernandes
Andrew M. Thompson
Daniele Castagnolo
William A. Denny
Jean L. Dos Santos
Published in:
Journal of Medicinal Chemistry, Issue 65, 2022, Page(s) 7489–7531, ISSN 0022-2623
Publisher:
American Chemical Society
DOI:
10.1021/acs.jmedchem.2c00227
Development of Novel Membrane Disrupting Lipoguanidine Compounds Sensitizing Gram-Negative Bacteria to Antibiotics
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Author(s):
Seong-Heun Kim
Charlotte K. Hind
Guilherme F. S. Fernandes
Jingyue Wu
Dorothy Semenya
Melanie Clifford
Caleb Marsh
Silvia Anselmi
A. James Mason
Kenneth D. Bruce
J. Mark Sutton
Daniele Castagnolo
Published in:
ACS Medicinal Chemistry Letters, 2024, ISSN 1948-5875
Publisher:
American Chemical Society
DOI:
10.1021/acsmedchemlett.3c00460