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Innovative Mechanochemical Processes to synthesize green ACTIVE pharmaceutical ingredients.

Publicaciones

Sustainable Beckmann Rearrangement using Bead-Milling Technology: The Route to Paracetamol

Autores: Geib, R.; Colacino, E.; Gremaud, L.
Publicado en: ChemSusChem, 2024, ISSN 1864-564X
Editor: Wiley-VCH GmbH, Weinheim
DOI: 10.1002/cssc.202301921

Green metrics in mechanochemistry

Autores: Fantozzi, Nicolas; Volle, Jean-Noël; Porcheddu, Andrea; Virieux, David; Garcia, Felipe; Colacino, Evelina
Publicado en: Chemical Society Reviews, Edición 52, 2023, ISSN 0306-0012
Editor: Royal Society of Chemistry
DOI: 10.1039/D2CS00997H

Scalability of Pharmaceutical Co-Crystal Formation by Mechanochemistry in Batch

Autores: Bodach, Alexander; PORTET, Anaïs; Winkelmann, Frederik; Bastian, Herrmann; Gallou, Fabrice; Ponnusamy, Ettigounder; VIRIEUX, David; Colacino, Evelina; Felderhoff, Michael
Publicado en: ChemSusChem, 2023, ISSN 1864-5631
Editor: Wiley-VCH GmbH
DOI: 10.1002/cssc.202301220

Protecting-Group-Free Mechanosynthesis of Amides from Hydroxycarboxylic Acids: Application to the Synthesis of Imatinib

Autores: Nikonovich, Tatsiana; Jarg, Tatsiana; Martõnova, Jevgenija; Kudrjašov, Artjom; Merzhyievskyi, Danylo; Kudrjašova, Marina; Gallou, Fabrice; Aav, Riina; Kananovich, Dzmitry
Publicado en: ChemRxiv, 2023, ISSN 2573-2293
Editor: ChemRxiv
DOI: 10.26434/chemrxiv-2023-d4nxn

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