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G-quadruplexes in the HIV-1 genome: novel targets for the development of selective antiviral drugs

CORDIS fournit des liens vers les livrables publics et les publications des projets HORIZON.

Les liens vers les livrables et les publications des projets du 7e PC, ainsi que les liens vers certains types de résultats spécifiques tels que les jeux de données et les logiciels, sont récupérés dynamiquement sur OpenAIRE .

Publications

G-quadruplex fluorescence sensing by core-extended naphthalene diimides

Auteurs: Zuffo Michela; Doria Filippo; Botti Silvia; Bergamaschi Greta; Freccero Mauro
Publié dans: Elsevier BVBiochimica et Biophysica Acta - General Subjects 2017
Identifiant permanent: Digital Object Identifier:10.1016/j.bbagen.2016.11.034; PubMed ID:27902935; Microsoft Academic Graph Identifier:2549108696; Handle:20.500.14243/402022; Handle:11571/1181013

Targeting of RET oncogene by naphthalene diimide-mediated gene promoter G-quadruplex stabilization exerts anti-tumor activity in oncogene-addicted human medullary thyroid cancer

Auteurs: Lopergolo, Alessia; Perrone, Rosalba; Tortoreto, Monica; Beretta, Giovanni L.; Zuco, Valentina; Borrello, Maria Grazia; Lanzi, Cinzia; Richter, Sara N.; Zaffaroni, Nadia; Folini, Marco; DORIA, FILIPPO; FRECCERO, MAURO
Publié dans: Impact Journals, LLCOncotarget 2016
Identifiant permanent: Digital Object Identifier:10.18632/oncotarget.10105; PubMed ID:27351133; PubMed Central ID:PMC5226536; Microsoft Academic Graph Identifier:2419736060; Handle:11571/1163802

Nucleolin stabilizes G-quadruplex structures folded by the LTR promoter and silences HIV-1 viral transcription

Auteurs: TOSONI, ELENA; FRASSON, ILARIA; SCALABRIN, MATTEO; PERRONE, ROSALBA; BUTOVSKAYA, ELENA; NADAI, MATTEO; PALU', GIORGIO; Fabris, Dan; RICHTER, SARA
Publié dans: Oxford University Press (OUP)Nucleic Acids Research 2015
Identifiant permanent: Digital Object Identifier:10.1093/nar/gkv897; PubMed ID:26354862; PubMed Central ID:PMC4605322; Microsoft Academic Graph Identifier:1862469243; Handle:11577/3168422

Naphthalene Diimide–Tetraazacycloalkane Conjugates Are G-Quadruplex-Based HIV-1 Inhibitors with a Dual Mode of Action

Auteurs: Matteo Nadai; Filippo Doria; Ilaria Frasson; Rosalba Perrone; Valentina Pirota; Greta Bergamaschi; Mauro Freccero; Sara N. Richter
Publié dans: American Chemical Society (ACS)ACS Infect Dis 2024
Identifiant permanent: Digital Object Identifier:10.1021/acsinfecdis.3c00453; PubMed ID:38175706; PubMed Central ID:PMC10862543; Handle:20.500.14243/509919; Handle:11571/1488018

Oxadiazole/Pyridine-Based Ligands: A Structural Tuning for Enhancing G-Quadruplex Binding

Auteurs: Filippo Doria; Valentina Pirota; Michele Petenzi; Marie-Paule Teulade-Fichou; Daniela Verga; Mauro Freccero
Publié dans: MDPI AGMolecules, Vol 23, Iss 9, p 2162 (2018) 2018
Identifiant permanent: Digital Object Identifier:10.3390/molecules23092162; PubMed ID:30154319; PubMed Central ID:PMC6225118; Microsoft Academic Graph Identifier:2889400821; Handle:11571/1231106

A Catalytic and Selective Scissoring Molecular Tool for Quadruplex Nucleic Acids

Auteurs: Matteo Nadai; Filippo Doria; Matteo Scalabrin; Valentina Pirota; Vincenzo Grande; Greta Bergamaschi; Valeria Amendola; Fernaldo Richtia Winnerdy; Anh Tuân Phan; Sara N. Richter; Mauro Freccero
Publié dans: American Chemical Society (ACS)Journal of the American Chemical Society 2018
Identifiant permanent: Digital Object Identifier:10.1021/jacs.8b05337; PubMed ID:30351011; PubMed Central ID:PMC6242190; Microsoft Academic Graph Identifier:2896466432; Handle:20.500.14243/345495; Handle:10356/139320; Handle:11571/1231186

A bimodal fluorescent and photocytotoxic naphthalene diimide for theranostic applications

Auteurs: Salvati Erica; Doria Filippo; Manoli Francesco; D'Angelo Carmen; Biroccio Annamaria; Freccero Mauro; Manet Ilse
Publié dans: Royal Society of Chemistry (RSC)info:cnr-pdr/source/autori:Salvati, Erica; Doria, Filippo; Manoli, Francesco;* D'Angelo, Carmen; Biroccio, Annamaria; Freccero, Mauro; Manet, Ilse*/titolo:A bimodal fluorescent and photocytotoxic naphthalene diimide for theranostic applications/doi:10.1039/c6ob00987e/rivista:Organic & biomolecular chemistry/anno:2016/pagina_da:7238/pagina_a:7249/intervallo_pagine:7238–7249/volume:14 2016
Identifiant permanent: Digital Object Identifier:10.1039/c6ob00987e; PubMed ID:27383473; Microsoft Academic Graph Identifier:2476808476; Handle:20.500.14243/354225; Handle:11571/1163304

Antiviral Activity of the G-Quadruplex Ligand TMPyP4 against Herpes Simplex Virus-1

Auteurs: Sara Artusi; Emanuela Ruggiero; Matteo Nadai; Beatrice Tosoni; Rosalba Perrone; Annalisa Ferino; Irene Zanin; Luigi Xodo; Louis Flamand; Sara N. Richter
Publié dans: MDPI AGVolume 13 2021
Identifiant permanent: Digital Object Identifier:10.3390/v13020196; PubMed ID:33525505; PubMed Central ID:PMC7911665; Microsoft Academic Graph Identifier:3123301455

Mapping and characterization of G-quadruplexes in Mycobacterium tuberculosis gene promoter regions

Auteurs: Perrone, Rosalba; Lavezzo, Enrico; Riello, Erika; Manganelli, Riccardo; PalÃ1, Giorgio; Toppo, Stefano; Provvedi, Roberta; Richter, Sara N.
Publié dans: Springer Science and Business Media LLCSci Rep 2017
Identifiant permanent: Digital Object Identifier:10.1038/s41598-017-05867-z; PubMed ID:28720801; PubMed Central ID:PMC5515968; Microsoft Academic Graph Identifier:2736256689; Handle:11577/3248797

The Oncogenic Signaling Pathways in BRAF-Mutant Melanoma Cells Are Modulated by Naphthalene Diimide-Like G-Quadruplex Ligands

Auteurs: Marta Recagni; Martina Tassinari; Filippo Doria; Graziella Cimino-Reale; Nadia Zaffaroni; Mauro Freccero; Marco Folini; Sara N. Richter
Publié dans: MDPI AGVolume 8 2019
Identifiant permanent: Digital Object Identifier:10.3390/cells8101274; PubMed ID:31635389; PubMed Central ID:PMC6830342; Microsoft Academic Graph Identifier:2980848506; Handle:11571/1351174

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