Publications Peer reviewed articles (13) Targeting MYC Proteins for Tumor Therapy Author(s): Elmar Wolf, Martin Eilers Published in: Annual Review of Cancer Biology, Issue 4/1, 2020, Page(s) 61-75, ISSN 2472-3428 Publisher: Annual Reviews DOI: 10.1146/annurev-cancerbio-030518-055826 NOXA expression drives synthetic lethality to RUNX1 inhibition in pancreatic cancer Author(s): Josefina Doffo, Stefanos A Bamopoulos, Hazal Köse, Felix Orben , Chuanbing Zang , Miriam Pons , Alexander T den Dekker , Rutger W W Brouwer, Apoorva Baluapuri , Stefan Habringer, Maximillian Reichert , Anuradha Illendula , Oliver H Krämer , Markus Schick, Elmar Wolf, Wilfred F J van IJcken, Irene Esposito, Ulrich Keller, Günter Schneider, Matthias Wirth Published in: Proceedings of the National Academy of Sciences of the United States of America, 2022, ISSN 0027-8424 Publisher: National Academy of Sciences DOI: 10.1073/pnas.2105691119 Generation of auxin inducible degron (AID) knock-in cell lines for targeted protein degradation in mammalian cells Author(s): Bikash Adhikari, Ashwin Narain, and Elmar Wolf Published in: Star Protocols, 2021, ISSN 2666-1667 Publisher: Cell Press Elsevier Inc. DOI: 10.1016/j.xpro.2021.100949 Novel, highly potent PROTACs targeting AURORA-A kinase Author(s): Jelena Bozilovic, Lorenz Eing , Benedict-Tilman Berger, Bikash Adhikari, Janik Weckesser, Nicola B. Berner d, Stephanie Wilhelm, Bernhard Kuster, Elmar Wolf, Stefan Knapp Published in: Current Research in Chemical Biology, 2022, ISSN 2666-2469 Publisher: Elsevier DOI: 10.1016/j.crchbi.2022.100032 MYC multimers shield stalled replication forks from RNA polymerase Author(s): Daniel Solvie, Apoorva Baluapuri, Leonie Uhl, Daniel Fleischhauer, Theresa Endres, Dimitrios Papadopoulos, Amel Aziba, Abdallah Gaballa, Ivan Mikicic, Ekaterina Isaakova, Celeste Giansanti, Jennifer Jansen, Marvin Jungblut, Teresa Klein, Christina Schülein-Völk, Hans Maric, Sören Doose, Markus Sauer, Petra Beli, Andreas Rosenwald, Matthias Dobbelstein, Elmar Wolf, Martin Eiles Published in: Nature, 2022, ISSN 0028-0836 Publisher: Nature Publishing Group DOI: 10.1038/s41586-022-05469-4 PROTAC-mediated degradation reveals a non-catalytic function of AURORA-A kinase Author(s): Bikash Adhikari, Jelena Bozilovic, Mathias Diebold, Jessica Denise Schwarz, Julia Hofstetter, Martin Schröder, Marek Wanior, Ashwin Narain, Markus Vogt, Nevenka Dudvarski Stankovic, Apoorva Baluapuri, Lars Schönemann, Lorenz Eing, Pranjali Bhandare, Bernhard Kuster, Andreas Schlosser, Stephanie Heinzlmeir, Christoph Sotriffer, Stefan Knapp, Elmar Wolf Published in: Nature Chemical Biology, Issue 16/11, 2020, Page(s) 1179-1188, ISSN 1552-4450 Publisher: Nature Publishing Group DOI: 10.1038/s41589-020-00652-y Target gene-independent functions of MYC oncoproteins Author(s): Apoorva Baluapuri, Elmar Wolf, Martin Eilers Published in: Nature Reviews Molecular Cell Biology, Issue 21/5, 2020, Page(s) 255-267, ISSN 1471-0072 Publisher: Nature Publishing Group DOI: 10.1038/s41580-020-0215-2 MYC Recruits SPT5 to RNA Polymerase II to Promote Processive Transcription Elongation Author(s): Apoorva Baluapuri, Julia Hofstetter, Nevenka Dudvarski Stankovic, Theresa Endres, Pranjali Bhandare, Seychelle Monique Vos, Bikash Adhikari, Jessica Denise Schwarz, Ashwin Narain, Markus Vogt, Shuang-Yan Wang, Robert Düster, Lisa Anna Jung, Jens Thorsten Vanselow, Armin Wiegering, Matthias Geyer, Hans Michael Maric, Peter Gallant, Susanne Walz, Andreas Schlosser, Patrick Cramer, Martin Eilers, El Published in: Molecular Cell, Issue 74/4, 2019, Page(s) 674-687.e11, ISSN 1097-2765 Publisher: Cell Press DOI: 10.1016/j.molcel.2019.02.031 Design, Synthesis, and Evaluation of WD-Repeat-Containing Protein 5 (WDR5) Degraders Author(s): Anja Dölle, Bikash Adhikari, Andreas Krämer, Janik Weckesser, Nicola Berner, Lena-Marie Berger, Mathias Diebold, Magdalena M. Szewczyk, Dalia Barsyte-Lovejoy, Cheryl H. Arrowsmith, Jakob Gebel, Frank Löhr, Volker Dötsch, Martin Eilers, Stephanie Heinzlmeir, Bernhard Kuster, Christoph Sotriffer, Elmar Wolf*, and Stefan Knapp* Published in: Journal of Medicinal Chemistry, 2021, ISSN 0022-2623 Publisher: American Chemical Society DOI: 10.1021/acs.jmedchem.1c00146 MondoA drives malignancy in B-ALL through enhanced adaptation to metabolic stress Author(s): Alexandra Sipol, Erik Hameister, Busheng Xue, Julia Hofstetter, Maxim Barenboim, Rupert Öllinger, Gaurav Jain, Carolin Prexler, Rebeca Alba Rubio, Michaela C. Baldauf, Davide G. Franchina, Andreas Petry, Juliane Schmäh, Uwe Thiel, Agnes Görlach, Gunnar Cario, Dirk Brenner, Günther H. S. Richter, Thomas G. P. Grünewald, Roland Rad, Elmar Wolf, Jürgen Ruland, Poul H. Sorensen, Stefan E. G. Bur Published in: BLOOD, 2021, ISSN 1528-0020 Publisher: American Society of Hematology DOI: 10.1182/blood.2020007932 The glycolytic enzyme ALDOA and the exon junction complex protein RBM8A are regulators of ribosomal biogenesis Author(s): Jessica Denise Schwarz, Sören Lukassen, Pranjali Bhandare, Lorenz Eing, Marteinn Thor Snaebjörnsson, Yiliam Cruz García, Jan Philipp Kisker, Almut Schulze and Elmar Wolf Published in: Frontiers in Cell and Developmental Biology, 2022, ISSN 2296-634X Publisher: Frontiers Media DOI: 10.3389/fcell.2022.954358 Tumor-Derived Lactic Acid Modulates Activation and Metabolic Status of Draining Lymph Node Stroma Author(s): Angela Riedel, Moutaz Helal, Luisa Pedro, Jonathan J. Swietlik, David Shorthouse, Werner Schmitz , Lisa Haas, Timothy Young, Ana S.H. da Costa, Sarah Davidson, Pranjali Bhandare, Elmar Wolf, Benjamin A. Hall, Christian Frezza, Thordur Oskarsson, and Jacqueline D. Shields Published in: CANCER IMMUNOLOGY RESEARCH, 2022, ISSN 2326-6066 Publisher: American Association for Cancer Research Inc. DOI: 10.1158/2326-6066.cir-21-0778 Targeted protein degradation reveals a direct role of SPT6 in RNAPII elongation and termination Author(s): Ashwin Narain, Pranjali Bhandare, Bikash Adhikari, Simone Backes, Martin Eilers, Lars Dö lken, Andreas Schlosser, Florian Erhard, Apoorva Baluapuri, and Elmar Wolf Published in: Molecular Cell, 2021, ISSN 1097-2765 Publisher: Cell Press DOI: 10.1016/j.molcel.2021.06.016 Searching for OpenAIRE data... There was an error trying to search data from OpenAIRE No results available