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From the understanding of KRAS-RAF membrane dynamics to new therapeutic strategies in cancer

Publicaciones

The phospholipid transporter PITPNC1 links KRAS to MYC to prevent autophagy in lung and pancreatic cancer

Autores: Entrialgo-Cadierno, Rodrigo; Cueto-Ureña, Cristina; Welch, Connor; Feliu, Iker; Macaya, Irati; Vera, Laura; Morales, Xabier; Michelina, Sandra Vietti; Scaparone, Pietro; Lopez, Ines; Darbo, Elodie; Erice, Oihane; Vallejo, Adrian; Moreno, Haritz; Goñi-Salaverri, Ainhoa; Lara-Astiaso, David; Halberg, Nils; Cortes-Dominguez, Ivan; Guruceaga, Elizabeth; Ambrogio, Chiara; Lecanda, Fernando; Vicent,
Publicado en: Molecular Cancer, Vol 22, Iss 1, Pp 1-23 (2023), Edición 2, 2023, ISSN 1476-4598
Editor: BioMed Central
DOI: 10.1186/s12943-023-01788-w

Structural model of a Ras-Raf signalosome

Autores: Mysore VP*, Zhou Z*, Ambrogio C*, Wang Q, Okoro J, Jänne PA, Westover KD, Shan Y, Shaw DE
Publicado en: Nature Structural and Molecular Biology, 2021, ISSN 1545-9993
Editor: Nature Publishing Group
DOI: 10.1038/s41594-021-00667-6

Concurrent inhibition of oncogenic and wild-type RAS-GTP for cancer therapy

Autores: Mallika Singh; Matthew Holderfield; Bianca Lee; Jingjing Jiang; Aidan Tomlinson; Kyle Seamon; Alessia Mira; Enricho Patrucco; Grace Goodhart; Julien Dilly; Yevgeniy Gindin; Nuntana Dinglasan; Ying Wang; Lick Pui Lai; Shurui Cai; Lingyan Jiang; Yu Yang; Nicole Nasholm; James Evans; Nilufar Montazer; Oliver Lai; Jade Shi; Ethan Ahler; Stephanie Chang; Anthony Salvador; Abby Marquez; Jim Cregg; Yang
Publicado en: Nature, Edición 1, 2024, ISSN 1476-4687
Editor: Nature Publishing Group
DOI: 10.21203/rs.3.rs-3122478/v1

Comparative Analysis and Isoform-Specific Therapeutic Vulnerabilities of KRAS Mutations in Non-Small Cell Lung Cancer

Autores: Biagio Ricciuti, Jieun Son, Jeffrey J Okoro, Alessia Mira, Enrico Patrucco, Yoonji Eum, Xinan Wang, Raymond Paranal, Haiyun Wang, Mika Lin, Heidi M Haikala, Jiaqi Li, Yue Xu, Joao Victor Alessi, Chhayheng Chhoeu, Amanda J Redig, Jens Köhler, Kshiti H Dholakia, Yunhan Chen, Elodie Richard, Marie-Julie Nokin, David Santamaria, Prafulla C Gokhale, Mark M Awad, Pasi A Jänne, Chiara Ambrogio
Publicado en: Clinical Cancer Research, 2022, ISSN 1078-0432
Editor: American Association for Cancer Research
DOI: 10.1158/1078-0432.ccr-21-2719

Biological and targeting differences between the rare KRAS A146T and canonical KRAS mutants in gastric cancer models

Autores: Elisabetta Puliga, Chiara De Bellis, Sandra Vietti Michelina, Tania Capeloa, Cristina Migliore, Claudia Orrù, Gian Luca Baiocchi, Giovanni De Manzoni, Filippo Pietrantonio, Rossella Reddavid, Uberto Fumagalli Romario, Chiara Ambrogio, Simona Corso, Silvia Giordano
Publicado en: Gastric Cancer, Edición 27, 2024, ISSN 1436-3305
Editor: Springer
DOI: 10.1007/s10120-024-01468-8

Novel RAF-directed approaches to overcome current clinical limits and block the RAS/RAF node

Autores: Rossella Scardaci, Ewa Berlinska, Pietro Scaparone, Sandra Vietti Michelina, Edoardo Garbo, Silvia Novello, David Santamaria, Chiara Ambrogio
Publicado en: Molecular Oncology, 2024, ISSN 1878-0261
Editor: FEBS PRESS
DOI: 10.1002/1878-0261.13605

Genomic Profiling Identifies Putative Pathogenic Alterations in NSCLC Brain Metastases

Autores: Marcin Nicoś, Luuk Harbers, Enrico Patrucco, Maximilian Kramer-Drauberg, Xiaolu Zhang 1 2 5 , Claudia Voena 4 , Anna Kowalczyk 6 7 , Aleksandra Bożyk 3 , Rafał Pęksa 7 8 , Bożena Jarosz 7 9 , Justyna Szumiło 10 , Michele Simonetti 1 2 , Monika Żuk 11 , Bartosz Wasąg 11 , Katarzyna Reszka 12 , Renata Duchnowska 7 13 , Janusz Milanowski 3 , Roberto Chiarle 4 14
Publicado en: JTO Clin Res Rep, Edición VOL 3 (12), 2022, ISSN 2666-3643
Editor: New York: Elsevier Inc.
DOI: 10.1016/j.jtocrr.2022.100435

Exploiting signaling rewiring in cancer cells with co‐existing oncogenic drivers

Autores: Roberto Chiarle; Chiara Ambrogio
Publicado en: Molecular Oncology, Vol 17, Iss 11, Pp 2215-2217 (2023), Edición 2, 2023, ISSN 1878-0261
Editor: Elsevier
DOI: 10.1002/1878-0261.13547

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