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Peptide-Drug Conjugates for Targeted Delivery in Tumor Therapy

Deliverables

International Network Symposium

International Network Symposium held

Summer School

Summer School held

Feature article on Peptide-Drug Conjugates

Feature article on Peptide-Drug Conjugates published in a popular scientific journal

Special issue on Peptide-Drug Conjugates

Special issue on Peptide-Drug Conjugates published in a scientific journal

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Completion of Website

Videos

Videos on ETN activities published by Beilstein TV

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Publications

Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α V β 3

Author(s): André Raposo Moreira Dias, Arianna Pina, Alberto Dal Corso, Daniela Arosio, Laura Belvisi, Luca Pignataro, Michele Caruso, Cesare Gennari
Published in: Chemistry - A European Journal, Issue 23/58, 2017, Page(s) 14410-14415, ISSN 0947-6539
DOI: 10.1002/chem.201703093

Tumor Targeting with an iso DGR-Drug Conjugate

Author(s): Simone Zanella, Simona Angerani, Arianna Pina, Paula López Rivas, Clelia Giannini, Silvia Panzeri, Daniela Arosio, Michele Caruso, Fabio Gasparri, Ivan Fraietta, Clara Albanese, Aurelio Marsiglio, Luca Pignataro, Laura Belvisi, Umberto Piarulli, Cesare Gennari
Published in: Chemistry - A European Journal, Issue 23/33, 2017, Page(s) 7910-7914, ISSN 0947-6539
DOI: 10.1002/chem.201701844

Convenient Preparation of 18F-Labeled Peptide Probes for Potential Claudin-4 PET Imaging

Author(s): Lucia Feni, M. Omrane, Moritz Fischer, Boris Zlatopolskiy, Bernd Neumaier, Ines Neundorf
Published in: Pharmaceuticals, Issue 10/4, 2017, Page(s) 99, ISSN 1424-8247
DOI: 10.3390/ph10040099

Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin–GnRH-III conjugates developed for targeted drug delivery

Author(s): Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, Viktor Farkas, László Buday, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Published in: Beilstein Journal of Organic Chemistry, Issue 14, 2018, Page(s) 756-771, ISSN 1860-5397
DOI: 10.3762/bjoc.14.64

Development of novel cyclic NGR peptide–daunomycin conjugates with dual targeting property

Author(s): Andrea Angelo Pierluigi Tripodi, Szilárd Tóth, Kata Nóra Enyedi, Gitta Schlosser, Gergely Szakács, Gábor Mező
Published in: Beilstein Journal of Organic Chemistry, Issue 14, 2018, Page(s) 911-918, ISSN 1860-5397
DOI: 10.3762/bjoc.14.78

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

Author(s): Lizeth Bodero, Paula López Rivas, Barbara Korsak, Torsten Hechler, Andreas Pahl, Christoph Müller, Daniela Arosio, Luca Pignataro, Cesare Gennari, Umberto Piarulli
Published in: Beilstein Journal of Organic Chemistry, Issue 14, 2018, Page(s) 407-415, ISSN 1860-5397
DOI: 10.3762/bjoc.14.29

Novel unit B cryptophycin analogues as payloads for targeted therapy

Author(s): Eduard Figueras, Adina Borbély, Mohamed Ismail, Marcel Frese, Norbert Sewald
Published in: Beilstein Journal of Organic Chemistry, Issue 14, 2018, Page(s) 1281-1286, ISSN 1860-5397
DOI: 10.3762/bjoc.14.109

Enhanced In Vitro Antitumor Activity of GnRH-III-Daunorubicin Bioconjugates Influenced by Sequence Modification

Author(s): Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, László Buday, János Gardi, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Published in: Pharmaceutics, Issue 10/4, 2018, Page(s) 223, ISSN 1999-4923
DOI: 10.3390/pharmaceutics10040223

Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and α V β 3 -Integrin Ligands for Tumor Targeting

Author(s): Paula López Rivas, Ivan Ranđelović, André Raposo Moreira Dias, Arianna Pina, Daniela Arosio, József Tóvári, Gábor Mező, Alberto Dal Corso, Luca Pignataro, Cesare Gennari
Published in: European Journal of Organic Chemistry, Issue 2018/23, 2018, Page(s) 2902-2909, ISSN 1434-193X
DOI: 10.1002/ejoc.201800447

In Vivo Antitumor Activity of a Novel Acetazolamide–Cryptophycin Conjugate for the Treatment of Renal Cell Carcinomas

Author(s): Samuele Cazzamalli, Eduard Figueras, Lilla Pethő, Adina Borbély, Christian Steinkühler, Dario Neri, Norbert Sewald
Published in: ACS Omega, Issue 3/11, 2018, Page(s) 14726-14731, ISSN 2470-1343
DOI: 10.1021/acsomega.8b02350

Cryptophycins: cytotoxic cyclodepsipeptides with potential for tumor targeting

Author(s): Christine Weiss, Eduard Figueras, Adina N. Borbely, Norbert Sewald
Published in: Journal of Peptide Science, Issue 23/7-8, 2017, Page(s) 514-531, ISSN 1075-2617
DOI: 10.1002/psc.3015

Characterization of a Cell-Penetrating Peptide with Potential Anticancer Activity

Author(s): Anja Gronewold, Mareike Horn, Ivan Ranđelović, Dr. József Tóvári, Sergio Muñoz Vázquez, Prof. Dr. Klaus Schomäcker, Prof. Dr. Ines Neundorf
Published in: ChemMedChem, Issue Januar 5, 2017, Volume 12, Issue 1, 2017, Page(s) 42–49, ISSN 1860-7187
DOI: 10.1002/cmdc.201600498

The Current Role of Cell-Penetrating Peptides in Cancer Therapy.

Author(s): Lucia Feni, Ines Neundorf
Published in: Peptides and Peptide-based Biomaterials and their Biomedical Applications. Advances in Experimental Medicine and Biology., Issue Vol 1030, 2017, Page(s) 279-295
DOI: 10.1007/978-3-319-66095-0_13