Peptide-Drug Conjugates for Targeted Delivery in Tumor Therapy

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Pubblicazioni

Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α V β 3

Autori: André Raposo Moreira Dias, Arianna Pina, Alberto Dal Corso, Daniela Arosio, Laura Belvisi, Luca Pignataro, Michele Caruso, Cesare Gennari
Pubblicato in: Chemistry - A European Journal, Numero 23/58, 2017, Pagina/e 14410-14415, ISSN 0947-6539
Editore: John Wiley & Sons Ltd.
DOI: 10.1002/chem.201703093

Tumor Targeting with an iso DGR-Drug Conjugate

Autori: Simone Zanella, Simona Angerani, Arianna Pina, Paula López Rivas, Clelia Giannini, Silvia Panzeri, Daniela Arosio, Michele Caruso, Fabio Gasparri, Ivan Fraietta, Clara Albanese, Aurelio Marsiglio, Luca Pignataro, Laura Belvisi, Umberto Piarulli, Cesare Gennari
Pubblicato in: Chemistry - A European Journal, Numero 23/33, 2017, Pagina/e 7910-7914, ISSN 0947-6539
Editore: John Wiley & Sons Ltd.
DOI: 10.1002/chem.201701844

Convenient Preparation of 18F-Labeled Peptide Probes for Potential Claudin-4 PET Imaging

Autori: Lucia Feni, M. Omrane, Moritz Fischer, Boris Zlatopolskiy, Bernd Neumaier, Ines Neundorf
Pubblicato in: Pharmaceuticals, Numero 10/4, 2017, Pagina/e 99, ISSN 1424-8247
Editore: Multidisciplinary Digital Publishing Institute (MDPI)
DOI: 10.3390/ph10040099

Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin–GnRH-III conjugates developed for targeted drug delivery

Autori: Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, Viktor Farkas, László Buday, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Pubblicato in: Beilstein Journal of Organic Chemistry, Numero 14, 2018, Pagina/e 756-771, ISSN 1860-5397
Editore: Beilstein-Institut
DOI: 10.3762/bjoc.14.64

Development of novel cyclic NGR peptide–daunomycin conjugates with dual targeting property

Autori: Andrea Angelo Pierluigi Tripodi, Szilárd Tóth, Kata Nóra Enyedi, Gitta Schlosser, Gergely Szakács, Gábor Mező
Pubblicato in: Beilstein Journal of Organic Chemistry, Numero 14, 2018, Pagina/e 911-918, ISSN 1860-5397
Editore: Beilstein-Institut
DOI: 10.3762/bjoc.14.78

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

Autori: Lizeth Bodero, Paula López Rivas, Barbara Korsak, Torsten Hechler, Andreas Pahl, Christoph Müller, Daniela Arosio, Luca Pignataro, Cesare Gennari, Umberto Piarulli
Pubblicato in: Beilstein Journal of Organic Chemistry, Numero 14, 2018, Pagina/e 407-415, ISSN 1860-5397
Editore: Beilstein-Institut
DOI: 10.3762/bjoc.14.29

Novel unit B cryptophycin analogues as payloads for targeted therapy

Autori: Eduard Figueras, Adina Borbély, Mohamed Ismail, Marcel Frese, Norbert Sewald
Pubblicato in: Beilstein Journal of Organic Chemistry, Numero 14, 2018, Pagina/e 1281-1286, ISSN 1860-5397
Editore: Beilstein-Institut
DOI: 10.3762/bjoc.14.109

Enhanced In Vitro Antitumor Activity of GnRH-III-Daunorubicin Bioconjugates Influenced by Sequence Modification

Autori: Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, László Buday, János Gardi, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Pubblicato in: Pharmaceutics, Numero 10/4, 2018, Pagina/e 223, ISSN 1999-4923
Editore: Multidisciplinary Digital Publishing Institute (MDPI)
DOI: 10.3390/pharmaceutics10040223

Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and α V β 3 -Integrin Ligands for Tumor Targeting

Autori: Paula López Rivas, Ivan Ranđelović, André Raposo Moreira Dias, Arianna Pina, Daniela Arosio, József Tóvári, Gábor Mező, Alberto Dal Corso, Luca Pignataro, Cesare Gennari
Pubblicato in: European Journal of Organic Chemistry, Numero 2018/23, 2018, Pagina/e 2902-2909, ISSN 1434-193X
Editore: John Wiley & Sons Ltd.
DOI: 10.1002/ejoc.201800447

In Vivo Antitumor Activity of a Novel Acetazolamide–Cryptophycin Conjugate for the Treatment of Renal Cell Carcinomas

Autori: Samuele Cazzamalli, Eduard Figueras, Lilla Pethő, Adina Borbély, Christian Steinkühler, Dario Neri, Norbert Sewald
Pubblicato in: ACS Omega, Numero 3/11, 2018, Pagina/e 14726-14731, ISSN 2470-1343
Editore: ACS Publications
DOI: 10.1021/acsomega.8b02350

Cryptophycins: cytotoxic cyclodepsipeptides with potential for tumor targeting

Autori: Christine Weiss, Eduard Figueras, Adina N. Borbely, Norbert Sewald
Pubblicato in: Journal of Peptide Science, Numero 23/7-8, 2017, Pagina/e 514-531, ISSN 1075-2617
Editore: John Wiley & Sons Inc.
DOI: 10.1002/psc.3015

Characterization of a Cell-Penetrating Peptide with Potential Anticancer Activity

Autori: Anja Gronewold, Mareike Horn, Ivan Ranđelović, Dr. József Tóvári, Sergio Muñoz Vázquez, Prof. Dr. Klaus Schomäcker, Prof. Dr. Ines Neundorf
Pubblicato in: ChemMedChem, Numero Januar 5, 2017, Volume 12, Numero 1, 2017, Pagina/e 42–49, ISSN 1860-7187
Editore: Wiley-VCH Verlag GmbH & Co. KGaA
DOI: 10.1002/cmdc.201600498

The Current Role of Cell-Penetrating Peptides in Cancer Therapy.

Autori: Lucia Feni, Ines Neundorf
Pubblicato in: Peptides and Peptide-based Biomaterials and their Biomedical Applications. Advances in Experimental Medicine and Biology., Numero Vol 1030, 2017, Pagina/e 279-295, ISBN 978-3-319-66094-3
Editore: Springer International Publishing
DOI: 10.1007/978-3-319-66095-0_13

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