Pubblicazioni Peer reviewed articles (9) Neutralizing the impact of the virulence factor LecA from Pseudomonas aeruginosa on human cells with new glycomimetic inhibitors Autori: Eva Zahorska, Francesca Rosato4,5+, Kai Stober4,5+, Sakonwan Kuhaudomlarp6-8, Joscha Meiers, Dirk Hauck, Dorina Reith4,5, Emilie Gillon6, Katharina Rox2,9, Anne Imberty6, Winfried Römer4,5,10*, Alexander Titz1-3* Pubblicato in: Angew. Chem. Int. Ed. Engl, 2022, ISSN 1433-7851 Editore: John Wiley & Sons Ltd. DOI: 10.1002/anie.202215535 Directing Drugs to Bugs: Antibiotic-Carbohydrate Conjugates Targeting Biofilm-Associated Lectins of Pseudomonas aeruginosa. Autori: Joscha Meiers; Eva Zahorska; Teresa Röhrig; Dirk Hauck; Stefanie Wagner; Alexander Titz Pubblicato in: United States, Numero 2, 2020, ISSN 0022-2623 Editore: American Chemical Society DOI: 10.1021/acs.jmedchem.0c00856 Nano-in-Microparticles for Aerosol Delivery ofAntibiotic-Loaded, Fucose-Derivatized, andMacrophage-Targeted Liposomes to Combat MycobacterialInfections: In Vitro Deposition, Pulmonary BarrierInteractions, and Targeted Delivery Autori: Benedikt C. Huck, Durairaj Thiyagarajan, Aghiad Bali, Annette Boese,Karen F. W. Besecke, Constantin Hozsa, Robert K. Gieseler, Marcus Furch,Cristiane Carvalho-Wodarz, Franziska Waldow, Dominik Schwudke, Olga Metelkina,Alexander Titz, Hanno Huwer, Konrad Schwarzkopf, Jessica Hoppstädter,Alexandra K. Kiemer, Marcus Koch, Brigitta Loretz,* and Claus-Michael Lehr Pubblicato in: Advanced Healthcare Materials, 2022, ISSN 2192-2640 Editore: John Wiley and Sons Ltd DOI: 10.1002/adhm.202102117 Targeting extracellular lectins of <i>Pseudomonas aeruginosa</i> with glycomimetic liposomes Autori: Olga Metelkina; Benedikt Huck; Jonathan S. O'Connor; Marcus Koch; Andreas Manz; Claus-Michael Lehr; Alexander Titz Pubblicato in: Crossref, Numero 1, 2022, ISSN 2050-7518 Editore: Royal Society of Chemistry DOI: 10.1039/d1tb02086b Discovery of <i>N</i>-β-<scp>l</scp>-Fucosyl Amides as High-Affinity Ligands for the <i>Pseudomonas aeruginosa</i> Lectin LecB Autori: Patrycja Mała; Eike Siebs; Joscha Meiers; Katharina Rox; Annabelle Varrot; Anne Imberty; Alexander Titz Pubblicato in: Crossref, Numero 4, 2022, ISSN 0022-2623 Editore: American Chemical Society DOI: 10.1021/acs.jmedchem.2c01373 A rapid synthesis of low-nanomolar divalent LecA inhibitors in four linear steps from D-galactose pentaacetate Autori: Eva Zahorska, Sakonwan Kuhaudomlarp, Saverio Minervini, Sultaan Yousaf, Martin Lepsik, Thorsten Kinsinger, Anna K. H. Hirsch, Anne Imberty and Alexander Titz Pubblicato in: ChemComm, 2020, ISSN 1364-548X Editore: Royal Chemical Society DOI: 10.1039/d0cc03490h Covalent Lectin Inhibition and Application in Bacterial Biofilm Imaging Autori: Stefanie Wagner, Dirk Hauck, Michael Hoffmann, Roman Sommer, Ines Joachim, Rolf Müller, Anne Imberty, Annabelle Varrot, Alexander Titz Pubblicato in: Angewandte Chemie International Edition, Numero 56/52, 2017, Pagina/e 16559-16564, ISSN 1433-7851 Editore: John Wiley & Sons Ltd. DOI: 10.1002/anie.201709368 Anti-biofilm Agents against Pseudomonas aeruginosa : A Structure–Activity Relationship Study of C -Glycosidic LecB Inhibitors Autori: Roman Sommer, Katharina Rox, Stefanie Wagner, Dirk Hauck, Sarah S. Henrikus, Shelby Newsad, Tatjana Arnold, Thomas Ryckmans, Mark Brönstrup, Anne Imberty, Annabelle Varrot, Rolf W. Hartmann, Alexander Titz Pubblicato in: Journal of Medicinal Chemistry, Numero 62/20, 2019, Pagina/e 9201-9216, ISSN 0022-2623 Editore: American Chemical Society DOI: 10.1021/acs.jmedchem.9b01120 Lectin-Targeted Prodrugs Activated by <i>Pseudomonas aeruginosa</i> for Self-Destructive Antibiotic Release Autori: Joscha Meiers; Katharina Rox; Alexander Titz Pubblicato in: Crossref, Numero 2, 2022, ISSN 0022-2623 Editore: American Chemical Society DOI: 10.1021/acs.jmedchem.2c01214 È in corso la ricerca di dati su OpenAIRE... Si è verificato un errore durante la ricerca dei dati su OpenAIRE Nessun risultato disponibile