Overlaid Transcriptional and Proteome Analyses Identify Mitotic Kinesins as Important Targets of Arylsulfonamide-Mediated RBM39 Degradation
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Autori:
Seemon Coomar;
Pedro Mota;
Alexander Penson;
Jürg Schwaller;
Omar Abdel-Wahab;
Dennis Gillingham
Pubblicato in:
Molecular Cancer Research, 2023, ISSN 1541-7786
Editore:
American Association for Cancer Research
DOI:
10.1158/1541-7786.mcr-22-0541
Repurposing the Damage Repair Protein Methyl Guanine Methyl Transferase as a Ligand Inducible Fusion Degron
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Autori:
Gosia M. Murawska, Caspar Vogel, Max Jan, Xinyan Lu, Matthias Schild, Mikolaj Slabicki, Charles Zou, Saule Zhanybekova, Manisha Manojkumar, Georg Petzold, Peter Kaiser, Nicolas Thomä, Benjamin Ebert, and Dennis Gillingham
Pubblicato in:
ACS Chemical Biology, Numero not yet known, 2022, Pagina/e not yet known, ISSN 1554-8929
Editore:
American Chemical Society
DOI:
10.1021/acschembio.1c00771
A high affinity pan-PI3K binding module supports selective targeted protein degradation of PI3Kα
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Autori:
Werner Theodor Jauslin, Matthias Schild, Thorsten Schaefer, Chiara Borsari, Clara Orbegozo, Lukas Bissegger, Saule Zhanybekova, Danilo Ritz, Alexander Schmidt, Matthias Wymann, Dennis Gillingham
Pubblicato in:
Chemical Science, Numero 15, 2024, Pagina/e 683-691, ISSN 2041-6520
Editore:
Royal Society of Chemistry
DOI:
10.1039/d3sc04629j