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A fully integrated, animal-free, end-to-end modelling approach to oral drug product development

Deliverables

Publications

Exploring the Cocrystal Landscape of Posaconazole by Combining High-Throughput Screening Experimentation with Computational Chemistry

Author(s): Matteo Guidetti, Rolf Hilfiker, Martin Kuentz, Annette Bauer-Brandl, Fritz Blatter
Published in: Crystal Growth & Design, Issue 23, 2, 2022, Page(s) 842-852, ISSN 1528-7483
Publisher: American Chemical Society
DOI: 10.1021/acs.cgd.2c01072

Microdialysis and nanofiltration allow to distinguish molecularly dissolved from colloid-associated drug concentrations during biomimetic dissolution testing of supersaturating formulations

Author(s): Florentin Lukas Holzem, Jeannine Petrig Schaffland, Martin Brandl, Annette Bauer-Brandl, Cordula Stillhart
Published in: European Journal of Pharmaceutical Sciences, Issue Volume 174, 1 July 2022, 2022, ISSN 0928-0987
Publisher: Elsevier BV
DOI: 10.1016/j.ejps.2022.106166

Biopredictive capability assessment of two dissolution/permeation assays, µFLUXTM and PermeaLoopTM, using supersaturating formulations of Posaconazole

Author(s): Florentin Lukas Holzem, Anika Weck, Jeannine Petrig Schaffland, Cordula Stillhart, Sandra Klein, Annette Bauer-Brandl, Martin Brandl
Published in: European Journal of Pharmaceutical Sciences, Issue 176, 2022, Page(s) 106260, ISSN 0928-0987
Publisher: Elsevier BV
DOI: 10.1016/j.ejps.2022.106260

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