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A fully integrated, animal-free, end-to-end modelling approach to oral drug product development

Rezultaty

Publikacje

Exploring the Cocrystal Landscape of Posaconazole by Combining High-Throughput Screening Experimentation with Computational Chemistry

Autorzy: Matteo Guidetti, Rolf Hilfiker, Martin Kuentz, Annette Bauer-Brandl, Fritz Blatter
Opublikowane w: Crystal Growth & Design, Numer 23, 2, 2022, Strona(/y) 842-852, ISSN 1528-7483
Wydawca: American Chemical Society
DOI: 10.1021/acs.cgd.2c01072

Polymer-embedded deep eutectic solvents (PEDES) as a novel bio-enabling formulation approach

Autorzy: Shaida Panbachi , Josef Beranek, Martin Kuentz
Opublikowane w: European Journal of Pharmaceutical Sciences, Numer Volume 186, 1 July 2023, 2023, ISSN 0928-0987
Wydawca: Elsevier BV
DOI: 10.1016/j.ejps.2023.106463

Projection of Target Drug Particle Size in Oral Formulations Using the Refined Developability Classification System (rDCS)

Autorzy: Kristian Beran; Eline Hermans; René Holm; Kia Sepassi; Jennifer Dressman
Opublikowane w: Pharmaceutics; Volume 15; Numer 7; Pages: 1909, Numer 1, 2023, ISSN 1999-4923
Wydawca: Multidisciplinary Digital Publishing Institute (MDPI)
DOI: 10.3390/pharmaceutics15071909

Microdialysis and nanofiltration allow to distinguish molecularly dissolved from colloid-associated drug concentrations during biomimetic dissolution testing of supersaturating formulations

Autorzy: Florentin Lukas Holzem, Jeannine Petrig Schaffland, Martin Brandl, Annette Bauer-Brandl, Cordula Stillhart
Opublikowane w: European Journal of Pharmaceutical Sciences, Numer Volume 174, 1 July 2022, 2022, ISSN 0928-0987
Wydawca: Elsevier BV
DOI: 10.1016/j.ejps.2022.106166

Biopredictive capability assessment of two dissolution/permeation assays, µFLUXTM and PermeaLoopTM, using supersaturating formulations of Posaconazole

Autorzy: Florentin Lukas Holzem, Anika Weck, Jeannine Petrig Schaffland, Cordula Stillhart, Sandra Klein, Annette Bauer-Brandl, Martin Brandl
Opublikowane w: European Journal of Pharmaceutical Sciences, Numer 176, 2022, Strona(/y) 106260, ISSN 0928-0987
Wydawca: Elsevier BV
DOI: 10.1016/j.ejps.2022.106260

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